BDBM50239382 Lidamidine

SMILES CN=C(N)NC(=O)Nc1c(C)cccc1C

InChI Key InChIKey=RRHJHSBDJDZUGL-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50239382   

TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50239382(Lidamidine)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hERG expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50239382(Lidamidine)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Cav1.2 expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50239382(Lidamidine)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetBile salt export pump(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50239382(Lidamidine)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human BSEP expressed in baculovirus transfected fall armyworm Sf21 cell membranes vesicles assessed as reduction in ATP-dependent [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2019
Entry Details Article
PubMed