BDBM82463 Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-amino*heptanoyl-L-Phe-)]::L-362,855::L-362855

SMILES C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)CCCCCCNC(=O)[C@H](Cc2ccccc2)NC1=O

InChI Key InChIKey=CDHQUESZSCDTRS-UHFFFAOYSA-N

Data  58 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 58 hits for monomerid = 82463   

TargetSomatostatin receptor type 4(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.00500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.670nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.670nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.670nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.760nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  1.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  1.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  1.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  1.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  1.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  2.04nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  2.04nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Mouse)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  2.96nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  4.36nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  4.36nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  4.37nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  5.12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  5.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  5.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  24.0nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  24.0nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Mouse)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  28.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Mouse)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  29nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  30.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Rat)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  49.0nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  49.0nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  51nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 4(Mouse)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  67.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  67.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  67.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  67.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  67.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  83.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Mouse)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  174nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  174nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82463(L-362855 | Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-...)
Affinity DataKi:  467nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
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