BDBM28799 2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)amino}ethyl)phenyl]sulfanyl}-2-methylpropanoic acid::CHEMBL278590::GW 9578::GW-9578::GW9578
SMILES CCCCCCCN(CCc1ccc(SC(C)(C)C(O)=O)cc1)C(=O)Nc1ccc(F)cc1F
InChI Key InChIKey=KYQNYMXQHLMADB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 34 hits for monomerid = 28799
Affinity DataEC50: 100nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibitory activity of compound against the binding of human Peroxisome proliferator activated receptor gamma was determinedMore data for this Ligand-Target Pair
Affinity DataEC50: 340nMAssay Description:Cotransfection activity of compound against human Peroxisome proliferator activated receptor alpha was determinedMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Agonist activity at PPARalpha ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at PPARdelta ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation...More data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Agonist activity at PPARgamma ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation...More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at Gal4-fused mouse PPARalphaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPARgammaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPARdeltaMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Cotransfection activity of compound against human Peroxisome proliferator activated receptor gamma was determinedMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARgammaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARdeltaMore data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Agonist activity at PPARalpha expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at PPARdelta expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 166nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Agonist activity at PPARgamma expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at human PPARalphaMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Agonist activity for Human PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Compound was tested for agonist activity on human Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor gamma-Gal4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor alpha-Gal4 chimeric receptor transfected CV-1 ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Compound was tested for agonist activity on human Peroxisome proliferator activated receptor gamma-Gal4 chimeric receptor in transfected CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Compound was tested for agonist activity on human Peroxisome proliferator activated receptor alpha-Gal4 chimeric receptor in transfected CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity for Human PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity for Human PPAR alpha receptor in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 78nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity for murine PPAR alpha receptor in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR delta ligand binding domainMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR gamma ligand binding domainMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR alpha ligand binding domainMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair