BDBM50070220 4-(6-Cyclopentyl-hex-3-ynyl)-1H-imidazole::CHEMBL274977::GT 2286

SMILES C(CC1CCCC1)C#CCCc1cnc[nH]1

InChI Key InChIKey=XFHACGZTJUJXHB-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50070220   

TargetHistamine H3 receptor(Rat)
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070220(GT 2286 | CHEMBL274977 | 4-(6-Cyclopentyl-hex-3-yn...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity at histamine H3 receptor in rat cortical membranes by [3H]Nalpha-methylhistamine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
Gliatech

Curated by PDSP Ki Database
LigandPNGBDBM50070220(GT 2286 | CHEMBL274977 | 4-(6-Cyclopentyl-hex-3-yn...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070220(GT 2286 | CHEMBL274977 | 4-(6-Cyclopentyl-hex-3-yn...)
Affinity DataKi:  0.950nMAssay Description:Antagonistic activity was evaluated against histamine H3 receptor using [3H]- N-alpha-methylhistamine as radioligand in experiment 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed