BDBM50280717 CHEMBL557974::CP-99711::N-[6,7-Dichloro-3-((E)-styryl)-quinoxalin-2-yl]-N,N',N'-trimethyl-propane-1,3-diamine; hydrochloride

SMILES CN(C)CCCN(C)c1nc2cc(Cl)c(Cl)cc2nc1\C=C\c1ccccc1

InChI Key InChIKey=FJJZLLDDYQTGGH-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50280717   

TargetGlucagon receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280717(N-[6,7-Dichloro-3-((E)-styryl)-quinoxalin-2-yl]-N,...)
Affinity DataIC50: 4.00E+3nMAssay Description:Tested against glucagon receptor for its ability to displace radiolabeled ([125I]-glucagon) in male Dawley rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetGlucagon receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280717(N-[6,7-Dichloro-3-((E)-styryl)-quinoxalin-2-yl]-N,...)
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [125I]-glucagon from GCGR in Sprague-Dawley rat liver assessed as decrease in glucagon-stimulated CAMP production incubated for 45 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed