BDBM50009453 CHEMBL259011::CHI-1043

SMILES COc1cccc2n(Cc3ccc(F)cc3)cc(C(=O)\C=C(/O)C(O)=O)c12

InChI Key InChIKey=GSMHULZNHJSXPP-UHFFFAOYSA-N

Data  11 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50009453   

TargetIntegrase(Human immunodeficiency virus type 1)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 140nMAssay Description:Inhibition of HIV-1 integrase strand transfer activity using 3'-end biotin labelled oligonucleotide/5'-end digoxigenin labelled oligonucleotide as su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 140nMAssay Description:Inhibition of HIV-1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 80nMAssay Description:Inhibition of HIV-1 integrase after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 110nMAssay Description:Inhibition of Human immunodeficiency virus 1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 140nMAssay Description:Inhibition of Human immunodeficiency virus 1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 80nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 140nMAssay Description:Inhibition of HIV1 integrase strand transferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 140nMAssay Description:Inhibition of HIV1 integrase strand transfer activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 80nMAssay Description:Inhibition of HIV1 integrase activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 140nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Central China Normal University

Curated by ChEMBL
LigandPNGBDBM50009453(CHEMBL259011 | CHI-1043)
Affinity DataIC50: 80nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed