BDBM50063839 BIM 23268::CHEMBL263606::H-cyclo[DCys-Phe-Phe-DTrp-Lys-Thr-Phe-DCys]-NH2

SMILES CC(O)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](N)CSSC[C@@H](NC(=O)[C@H](Cc2ccccc2)NC1=O)C(N)=O

InChI Key InChIKey=JNMPZUZCPFIJGJ-UHFFFAOYSA-N

Data  18 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 18 hits for monomerid = 50063839   

TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Mouse)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  1.49nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  2.18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Rat)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Mouse)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  15.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  15.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  16.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  16.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  18.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  18.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  61.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  61.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  101nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  174nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(CHEMBL263606 | BIM 23268 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  582nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed