BDBM93224 Kinase inhibitor, A1

SMILES CC1CN(CC(C)O1)c1nc2ccccn2c(=O)c1N

InChI Key InChIKey=GWZYDSKWIQPDBX-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 93224   

TargetCasein kinase II subunit alpha(Human)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 1.80E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 3(Human)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 2.10E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 1.96E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Chicken)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 9.70E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetSRSF protein kinase 1(Human)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 1.14E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed