BDBM754247 5-cyclopropyl-2-(4,4- difluoroazepan-1-yl)- N-(3-sulfamoyl- phenyl)nicotinamide::US12344595, Example 163

SMILES NS(=O)(=O)c1cccc(NC(=O)c2cc(C3CC3)cnc2N2CCCC(F)(F)CC2)c1

InChI Key

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 754247   

TargetSodium channel protein type 10 subunit alpha(Human)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 754247BDBM754247(5-cyclopropyl-2-(4,4- difluoroazepan-1-yl)- N-(3-s...)
Affinity DataIC50: 7.30nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent