BDBM752509 US20250197406, Example 100

SMILES CSCC(=O)Nc4cn3cc(c1c(Cl)c(F)c(NC(C)C)c2[nH]ncc12)ncc3n4

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 752509   

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
1ST Biotherapeutics

US Patent
LigandPNGBDBM752509(US20250197406, Example 100)
Affinity DataIC50: 100nMAssay Description:HPK1 kinase activity was measured by Promega's ADP-Glo™ kinase assay. In this assay, 5 ng of recombinant human HPK1 (signalchem) is incubated wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent