BDBM748916 US20250188078, Ref. PA78

SMILES CN(c1ccc(-c2nc(C(=O)O)cc3c2[nH]c2ccccc23)c(F)c1)S(=O)(=O)c1ccccc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 748916   

TargetCullin-4A/DNA damage-binding protein 1(Human)
Cornell University

US Patent
LigandPNGBDBM748916(US20250188078, Ref. PA78)
Affinity DataIC50: 840nMAssay Description:The means the half maximal inhibitory concentration of compound that inhibits CUL4A and DDB1-BPB binding. Our lab established and optimized 384 well-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
US Patent

TargetCullin-4A/DNA damage-binding protein 1(Human)
Cornell University

US Patent
LigandPNGBDBM748916(US20250188078, Ref. PA78)
Affinity DataKd:  3.44E+3nMAssay Description:To assess the interaction between DDB1-BPB and compounds, a multi-parametric SPR instrument (BioRad ProteON XPR360) was used. DDB1-BPB was immobilize...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
US Patent