BDBM748458 US20250188030, Compound C40

SMILES CC(C)S(=O)(=O)NC(=O)Cc1ccc(O[C@@H]2CC[C@@H](NC(=O)[C@]3(F)CNC4(CCC4)C3)C2)c(-c2cccc(F)c2C2CCC2)c1

InChI Key InChIKey=RVZBXBUXJSRYKX-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 748458   

TargetHistone acetyltransferase KAT2A(Human)
Pfizer

US Patent
LigandPNGBDBM748458(US20250188030, Compound C40)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT2B(Human)
Pfizer

US Patent
LigandPNGBDBM748458(US20250188030, Compound C40)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/7/2025
Entry Details
Go to US Patent