BDBM730933 (stereospecific Procedure): N-{6-[(3-cyclopropyl-1 H-pyrazol-5-yl)amino]-5-methoxy-1,2-benzoxazol-3-yl}-4-[(2S)-1,4-dioxan-2-yl]-2,6-dimethoxybenzene-1-sulfonamide::US20250122183, Example 146

SMILES COc1cc2c(NS(=O)(=O)c3c(OC)cc([C@H]4COCCO4)cc3OC)noc2cc1Cc1cc(C2CC2)n[nH]1

InChI Key InChIKey=OIJIORLVSSKPSQ-UHFFFAOYSA-N

Data  6 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 730933   

TargetHistone acetyltransferase KAT6A(Human)
Pfizer

US Patent
LigandPNGBDBM730933((stereospecific Procedure): N-{6-[(3-cyclopropyl-1...)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
Go to US Patent

LigandPNGBDBM730933((stereospecific Procedure): N-{6-[(3-cyclopropyl-1...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT7/Peregrin(Human)
Pfizer

US Patent
LigandPNGBDBM730933((stereospecific Procedure): N-{6-[(3-cyclopropyl-1...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
Go to US Patent

LigandPNGBDBM730933((stereospecific Procedure): N-{6-[(3-cyclopropyl-1...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT5(Human)
Pfizer

US Patent
LigandPNGBDBM730933((stereospecific Procedure): N-{6-[(3-cyclopropyl-1...)
Affinity DataKi:  31.4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT8(Human)
Pfizer

US Patent
LigandPNGBDBM730933((stereospecific Procedure): N-{6-[(3-cyclopropyl-1...)
Affinity DataKi:  865nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
Go to US Patent