BDBM723998 US20250064791, Compound Rosiglitazone

SMILES CN(CCOc1ccc(CC2SC(=O)NC2=O)cc1)c1ccccn1

InChI Key InChIKey=YASAKCUCGLMORW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 723998   

TargetMitochondrial pyruvate carrier 1/2(Human)
Minoryx Therapeutics

US Patent
LigandPNGBDBM723998(US20250064791, Compound Rosiglitazone)
Affinity DataIC50: 2.00E+3nMAssay Description:The MPC is a heterodimer composed of two subunits, MPC1 and MPC2. MPC1 and MPC2 interact to form an active carrier. In the assay, MPC2 was fused to R...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/29/2025
Entry Details
Go to US Patent