BDBM716530 N-((3R,5S)-5-((1H-Pyrazol-1-yl)methyl)-1-cyanopyrrolidin-3-yl)-6-(1H-indazol-4-yl)nicotinamide::US20250034122, Example 52

SMILES N#CN1C[C@H](NC(=O)c2ccc(-c3cccc4[nH]ncc34)nc2)C[C@H]1Cn1cccn1

InChI Key InChIKey=BLRGJXLUAARVPL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 716530   

TargetUbiquitin carboxyl-terminal hydrolase 30(Human)
Mission Therapeutics

US Patent
LigandPNGBDBM716530(N-((3R,5S)-5-((1H-Pyrazol-1-yl)methyl)-1-cyanopyrr...)
Affinity DataIC50: 15nMAssay Description:Dilution plates were prepared at 21 times the final concentration (2100 μM for a final concentration of 100 μM) in 50% DMSO in a 96-well polypropylen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
Go to US Patent