BDBM713969 US12202839, Compound 9p

SMILES CN1C(=O)C(=N)c2sc(-c3ccccc3)cc2C1=O

InChI Key InChIKey=IGPZTAJCUQIMOK-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 713969   

TargetProtein tyrosine phosphatase type IVA 3(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713969(US12202839, Compound 9p)
Affinity DataIC50: 48.9nMAssay Description:Table 2: Recombinant human PTP4A3 phosphatase was used and the enzymatic assay was performed as previously described,20 except that it was fully auto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetProtein tyrosine phosphatase type IVA 1 (PTP4A1)(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713969(US12202839, Compound 9p)
Affinity DataIC50: 133nMAssay Description:Table 4: In Vitro Biochemical Analysis of PTP4A Inhibition. Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black sma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetProtein tyrosine phosphatase type IVA 2 (PTP4A2)(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713969(US12202839, Compound 9p)
Affinity DataIC50: 264nMAssay Description:Table 4: In Vitro Biochemical Analysis of PTP4A Inhibition. Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black sma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetProtein tyrosine phosphatase type IVA 3(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713969(US12202839, Compound 9p)
Affinity DataIC50: 86nMAssay Description:Table 4: In Vitro Biochemical Analysis of PTP4A Inhibition. Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black sma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetProtein tyrosine phosphatase type IVA 3(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713969(US12202839, Compound 9p)
Affinity DataIC50: 48.9nMAssay Description:Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black small volume microtiter plates, as previously described using r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

TargetProtein tyrosine phosphatase type IVA 1 (PTP4A1)(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713969(US12202839, Compound 9p)
Affinity DataIC50: 133nMAssay Description:Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black small volume microtiter plates, as previously described using r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

TargetProtein tyrosine phosphatase type IVA 2 (PTP4A2)(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713969(US12202839, Compound 9p)
Affinity DataIC50: 264nMAssay Description:Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black small volume microtiter plates, as previously described using r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

TargetProtein tyrosine phosphatase type IVA 3(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713969(US12202839, Compound 9p)
Affinity DataIC50: 86nMAssay Description:Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black small volume microtiter plates, as previously described using r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent