BDBM708490 N-methyl-4-(3-(2-methyl- 5-((3- (trifluoromethyl)phenyl) carbamoyl)phenyl)pyrrolidin- 1-yl)picolinamide::US20240425482, Example 1

SMILES CNC(=O)c4cc(N3CCC(c2cc(C(=O)Nc1cccc(C(F)(F)F)c1)ccc2C)C3)ccn4

InChI Key InChIKey=ZCNJZWNALSVNKH-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 708490   

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chiesi Farmaceutici

US Patent
LigandPNGBDBM708490(N-methyl-4-(3-(2-methyl- 5-((3- (trifluoromethyl)p...)
Affinity DataKi: <10nMAssay Description:DDR1 and DDR2 binding assays were performed using Life Technologies LanthaScreen™ Europium Kinase Binding assay. The compounds were incubated with 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/7/2025
Entry Details
Go to US Patent

TargetDiscoidin domain-containing receptor 2(Human)
Chiesi Farmaceutici

US Patent
LigandPNGBDBM708490(N-methyl-4-(3-(2-methyl- 5-((3- (trifluoromethyl)p...)
Affinity DataKi: <10nMAssay Description:DDR1 and DDR2 binding assays were performed using Life Technologies LanthaScreen™ Europium Kinase Binding assay. The compounds were incubated with 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/7/2025
Entry Details
Go to US Patent