BDBM703751 (2S)-4-[3-fluoro-5- isobutyl-2-(2H- tetrazol-5-yl)phen- yl]-2-methyl-1-[(3- methyl-2-pyridyl)- methyl]piperazine::US20240368133, Compound A-228

SMILES Cc1cccnc1CN1CCN(c2cc(CC(C)C)cc(F)c2-c2nn[nH]n2)C[C@@H]1C

InChI Key InChIKey=OHDGYZFWUNUEDU-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 703751   

TargetType-2 angiotensin II receptor/Low affinity immunoglobulin epsilon Fc receptor(Human)
Confo Therapeutics

US Patent

LigandBDBM703751((2S)-4-[3-fluoro-5- isobutyl-2-(2H- tetrazol-5-yl)...)Copy SMILESCopy InChI

Affinity DataIC50: 14.9nMAssay Description:All synthesized ligands were evaluated in a radioligand assay by displacing 125I-[Sar1, Ile8]-Angiotensin II (Perkin Elmer, NEX248050UC) from human A...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
3/14/2025
Entry Details
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