BDBM702991 US20240366807, Compound 7290B

SMILES CB(O)[C@@H]1CCCN1C(=O)[C@@H](C)NC(=O)c1ccc(NCC(=O)CCc2ccc3n2[B-](F)(F)N2C(=C3)C(C)=CC2C)nc1

InChI Key InChIKey=FIVRVNZRLVKDRB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 702991   

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702991(US20240366807, Compound 7290B)
Affinity DataIC50: 13.9nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent