BDBM701212 1-[(4-cyclopropylphenyl)-methyl-carbamoyl]-4- [2-oxo-2-(N-tetrahydropyran-3- ylanilino)ethyl]piperidine-4-carboxylic acid::US12122750, Example 45B

SMILES CN(C(=O)N1CCC(CC(=O)N(c2ccccc2)C2CCCOC2)(C(=O)O)CC1)c1ccc(C2CC2)cc1

InChI Key InChIKey=GUSARVKGGSOURP-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 701212   

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM701212(1-[(4-cyclopropylphenyl)-methyl-carbamoyl]-4- [2-o...)
Affinity DataKi:  2.68nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
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Date in BDB:
2/24/2025
Entry Details
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