BDBM698782 US20240317755, Compound L015

SMILES Fc1ccc(C(=O)c2cnc3CN(CCn23)c2cn[nH]c(=O)c2Cl)c(c1)C(F)(F)F

InChI Key InChIKey=QKIXSAQMRMZSBN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 698782   

TargetShort transient receptor potential channel 5(Human)
Wuhan LL Science and Technology Development Co.

US Patent
LigandPNGBDBM698782(US20240317755, Compound L015)
Affinity DataIC50: 11.5nMAssay Description:TRPC5 is a type of non-selective cation channel with permeability to calcium ions. Therefore, TRPC5 agonist Englerin A (EA) and TRPC5 inhibitor Pico1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
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