BDBM689586 US12054502, Compound Bestazomib

SMILES CC(C)CC(NC(=O)C(O)C(N)Cc1ccccc1)B1OC(=O)C(CC(O)=C)(CC(O)=O)O1

InChI Key InChIKey=RJJQJNNPKHVRNV-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 689586   

TargetAminopeptidase N(Human)
Shandong Hubble Kisen Biological Technonlogy Co.

US Patent
LigandPNGBDBM689586(US12054502, Compound Bestazomib)
Affinity DataIC50: 2.14E+3nMAssay Description:Aminopeptidase N interacts with its commercial substrate L-leucyl p-nitroaniline (purchased from Sigma) to produce p-nitroaniline that is absorbed at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2024
Entry Details
Go to US Patent

TargetAminopeptidase N(Human)
Shandong Hubble Kisen Biological Technonlogy Co.

US Patent
LigandPNGBDBM689586(US12054502, Compound Bestazomib)
Affinity DataIC50: 3.87E+3nMAssay Description:Aminopeptidase N interacts with its commercial substrate L-leucyl p-nitroaniline (purchased from Sigma) to produce p-nitroaniline that is absorbed at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2024
Entry Details
Go to US Patent