BDBM683187 4-(5-(4 (dimethylamino) piperidin-1-yl)-8- (3-hydroxy-4- methoxyphenyl) imidazolo[1,2-c] pyrimidin-7-yl)-2- fluorobenzonitrile::US20240216357, Example 140

SMILES COc1ccc(cc1O)-c1c(nc(N2CCC(CC2)N(C)C)n2ccnc12)-c1ccc(C#N)c(F)c1

InChI Key InChIKey=DFOSQRYPZVYYPV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 683187   

TargetLysine-specific histone demethylase 1A(Human)
Sichuan Huiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM683187(US20240216357, Example 140 | 4-(5-(4 (dimethylamin...)
Affinity DataIC50: 0.400nMAssay Description:The effects of compounds on LSD1 enzyme activity are detected by an HTRF technology to evaluate their inhibition levels on LSD1 enzyme activity. Firs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2024
Entry Details
Go to US Patent