BDBM681938 US20240199649, Compound 214::US20240199649, Compound 382

SMILES CNc1nc(N[C@@H]2CCN(C)CC2(F)F)nn2ccc(-c3ccc4nc(C)n(CC(F)F)c4n3)c12

InChI Key InChIKey=SWPTWYNIHDNQQB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 681938   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Biosplice Therapeutics

US Patent
LigandPNGBDBM681938(US20240199649, Compound 382 | US20240199649, Compo...)
Affinity DataIC50: 1.10nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Division ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Biosplice Therapeutics

US Patent
LigandPNGBDBM681938(US20240199649, Compound 382 | US20240199649, Compo...)
Affinity DataIC50: 3.30nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Division ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent