BDBM667886 US20240122941, Compound 19

SMILES CCn1ncc(CN(C)C(=O)c2cc(nc3ccc(Cl)cc23)-c2ccc(NC3CN(C)C3)c(C)n2)c1C

InChI Key InChIKey=GYCCIEWETQNUJP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 667886   

TargetHistone acetyltransferase p300(Human)
National Cancer Center

US Patent
LigandPNGBDBM667886(US20240122941, Compound 19)
Affinity DataIC50: 17nMAssay Description:SensoLyte HAT (p300) Assay Kit (ANASPEC, AS-72172) was used to assess the HAT activity inhibiting capability of a HAT inhibitor. Specifically, 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2024
Entry Details
Go to US Patent