BDBM667882 US20240122941, Compound 16

SMILES CNC(=O)Nc1ccc2c(CC[C@]22OC(=O)N(CC(=O)N(Cc3ccc(F)cc3)C(C)C(F)(F)F)C2=O)c1

InChI Key InChIKey=VRVJKILQRBSEAG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 667882   

TargetHistone acetyltransferase p300(Human)
National Cancer Center

US Patent
LigandPNGBDBM667882(US20240122941, Compound 16)
Affinity DataIC50: 250nMAssay Description:SensoLyte HAT (p300) Assay Kit (ANASPEC, AS-72172) was used to assess the HAT activity inhibiting capability of a HAT inhibitor. Specifically, 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2024
Entry Details
Go to US Patent