BDBM667878 US20240122941, Compound 14

SMILES CC(N(Cc1ccc(F)cc1)C(=O)CN1C(=O)N[C@]2(CCc3cc(ccc23)-c2cnn(C)c2)C1=O)C(F)(F)F

InChI Key InChIKey=IBWWGICKBQHEBM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 667878   

TargetHistone acetyltransferase p300(Human)
National Cancer Center

US Patent
LigandPNGBDBM667878(US20240122941, Compound 14)
Affinity DataIC50: 70nMAssay Description:SensoLyte HAT (p300) Assay Kit (ANASPEC, AS-72172) was used to assess the HAT activity inhibiting capability of a HAT inhibitor. Specifically, 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2024
Entry Details
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