BDBM667873 US20240122941, Compound 5

SMILES FC(F)Oc1ccc(cc1)C1(CCC(F)(F)CC1)C(=O)N1CC(F)CC1C(=O)Nc1ccc2[nH]ncc2n1

InChI Key InChIKey=IGBIPTRCWSVZCO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 667873   

TargetHistone acetyltransferase p300(Human)
National Cancer Center

US Patent
LigandPNGBDBM667873(US20240122941, Compound 5)
Affinity DataIC50: 100nMAssay Description:SensoLyte HAT (p300) Assay Kit (ANASPEC, AS-72172) was used to assess the HAT activity inhibiting capability of a HAT inhibitor. Specifically, 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2024
Entry Details
Go to US Patent