BDBM667111 4-{7-[2-fluoro-5-(propan-2- yl)phenyl]-1H,2H,3H- pyrido[3,4-b][1,4]oxazin-1- yl}pyridin-2-amine::US20240116947, Example 13

SMILES CC(C)c1ccc(F)c(c1)-c1cc2N(CCOc2cn1)c1ccnc(N)c1

InChI Key InChIKey=DETKDYNFOUZRQO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 667111   

TargetTGF-beta receptor type-1(Human)
Chiesi Farmaceutici

US Patent
LigandPNGBDBM667111(US20240116947, Example 13 | 4-{7-[2-fluoro-5-(prop...)
Affinity DataIC50: 3nMAssay Description:The enzymatic activity of compounds of the present invention was monitored measuring the formation of ADP using the ADP-GLO Kinases assay. Following ...More data for this Ligand-Target Pair
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Date in BDB:
6/29/2024
Entry Details
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