BDBM664724 (R)-7-(3-amino-4-(2,4,5-trifluorophenyl)butanoyl)- 3-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,5- a]pyrazine-1-carboxylic acid::US20240115577, Compound 26

SMILES N[C@@H](CC(=O)N1CCn2c(C1)c(nc2C(F)(F)F)C(O)=O)Cc1cc(F)c(F)cc1F

InChI Key InChIKey=WJYKFSARHGEGEV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 664724   

TargetDipeptidyl peptidase 4(Human)
THE SCRIPPS RESEARCH INSTITUTE

US Patent
LigandPNGBDBM664724((R)-7-(3-amino-4-(2,4,5-trifluorophenyl)butanoyl)-...)
Affinity DataIC50: 0.800nMAssay Description:Human DPP4 activity assay data were obtained using a DPP4 Activity Assay Kit (Sigma-Aldrich, MAK088) according to the manufacturer's instructions...More data for this Ligand-Target Pair
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Date in BDB:
6/29/2024
Entry Details
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