BDBM661951 2-fluoro-4-(6-(1-methyl-1H-indazol-5-yl)- 3-((1-methylpiperidin-4-yl)methyl)-3H- imidazo[4,5-c]pyridin-7-yl)benzonitrile::US11944614, Compound 1

SMILES CNc1ccc(cc1C=N)-c1ncc2n(CC3CCN(C)CC3)cnc2c1-c1ccc(C#N)c(F)c1

InChI Key InChIKey=FLLYUSOFSNJOHN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 661951   

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandPNGBDBM661951(2-fluoro-4-(6-(1-methyl-1H-indazol-5-yl)- 3-((1-me...)
Affinity DataIC50: 40.1nMAssay Description:Enzymatic activity was assessed using the AlphaLISA technology from Perkin Elmer Life Sciences (Waltham, Mass.). 2.5 μL of compound solution and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2024
Entry Details
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