BDBM661372 US20240101559, Compound I-11

SMILES CN1CCC(CC1)Oc1ccc(Nc2nc3ccc(Oc4ccnc(NC(C)=O)c4)c4CCCn2c34)cc1C(F)(F)F

InChI Key InChIKey=NITZRVYMZIJERO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 661372   

TargetTyrosine-protein kinase JAK2(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM661372(US20240101559, Compound I-11)
Affinity DataIC50: 3.68E+3nMAssay Description:The JAK2 Z-Lyte biochemical assay was performed according to manufacturer's instructions (Life Technologies).More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2024
Entry Details
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