BDBM661043 N-(5-(((4-(1H-Pyrrolo[2,3-b]pyridin-2-yl)pyridin-2-yl)methyl)amino)-2-fluorophenyl)-2-phenylacetamide::US20240101538, Compound 18c

SMILES Fc1ccc(NCc2cc(ccn2)-c2cc3cccnc3[nH]2)cc1NC(=O)Cc1ccccc1

InChI Key InChIKey=SGKPVKAUCKPMFQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 661043   

TargetAurora kinase A(Human)
Eberhard Karls Universitat Tubingen

US Patent
LigandPNGBDBM661043(US20240101538, Compound 18c | N-(5-(((4-(1H-Pyrrol...)
Affinity DataIC50: 1.00E+4nMAssay Description:To measure the effect of the compounds on the activity of AURKA, the IC50 of the compounds was determined with the ADP-Glo Kinase Assay (Promega, V91...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2024
Entry Details
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