BDBM659471 US20240092770, Compound 128::US20240092770, Compound 73

SMILES CCN(CC)C(=O)c1csc(n1)S(=O)(=O)Nc1ccc(C)c2c(c[nH]c12)C#N

InChI Key InChIKey=YMEQSKFNNSFAMH-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 659471   

TargetRNA-binding protein 39 [150-331]/DDB1- and CUL4-associated factor 15(Human)
Recursion Pharmaceuticals

US Patent
LigandPNGBDBM659471(US20240092770, Compound 73 | US20240092770, Compou...)
Affinity DataEC50:  738nMAssay Description:A TR-FRET assay was used to assess the effect of compounds disclosed herein on the interaction between RBM39 and the DCAF15 complex. Test compounds w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2024
Entry Details
Go to US Patent

TargetRNA-binding protein 39 [150-331]/DDB1- and CUL4-associated factor 15(Human)
Recursion Pharmaceuticals

US Patent
LigandPNGBDBM659471(US20240092770, Compound 73 | US20240092770, Compou...)
Affinity DataEC50:  650nMAssay Description:A TR-FRET assay was used to assess the effect of compounds disclosed herein on the interaction between RBM39 and the DCAF15 complex. Test compounds w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2024
Entry Details
Go to US Patent