BDBM652419 US20240059682, Example 26
SMILES COc1nc2ccc(Oc3c(Cl)cc(cc3Cl)-n3nc(C#N)c(=O)[nH]c3=O)cc2n1C12CC(C1)C2
InChI Key InChIKey=NUCMFBMZGUIXNG-UHFFFAOYSA-N
Data 2 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 652419
TargetRetinoic acid receptor RXR-alpha/Thyroid hormone receptor beta(Human)
Terns Pharmaceuticals
US Patent
Terns Pharmaceuticals
US Patent
Affinity DataEC50: 1.26E+3nMAssay Description:Test compounds were prepared as 10 mM DMSO stock solutions. The stock solution (45 uL) was transferred to a 384-well assay plate, and 3-fold, 10-poin...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/Thyroid hormone receptor alpha(Human)
Terns Pharmaceuticals
US Patent
Terns Pharmaceuticals
US Patent
Affinity DataEC50: 2.50E+3nMAssay Description:Test compounds were prepared as 10 mM DMSO stock solutions. The stock solution (45 uL) was transferred to a 384-well assay plate, and 3-fold, 10-poin...More data for this Ligand-Target Pair