BDBM645385 N-(4-{[6-(5-chloro-2- fluorophenyl)pyridazin-4- ylamino}pyridin-2- yl)cyclopropanecarboxamide::US20240018122, Example 7

SMILES Fc1ccc(Cl)cc1-c1cc(Nc2ccnc(NC(=O)C3CC3)c2)cnn1

InChI Key InChIKey=GHYLVDJWXQEOCX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 645385   

TargetTGF-beta receptor type-1(Human)
Chiesi Farmaceutici

US Patent
LigandPNGBDBM645385(US20240018122, Example 7 | N-(4-{[6-(5-chloro-2- f...)
Affinity DataIC50: 1nMAssay Description:The enzymatic activity of compounds of the present invention was monitored measuring the formation of ADP using the ADP-GLO Kinases assay. Following ...More data for this Ligand-Target Pair
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Date in BDB:
3/13/2024
Entry Details
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