BDBM640925 (R)-4-(8-(3-aminopiperidin-1-yl)-3-(6-fluoro-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)imidazo[1,2-a]pyrazin-2-yl)-2-fluorobenzonitrile::US20230399332, Compound 30

SMILES Cn1nnc2cc(-c3c(nc4c(nccn34)N3CCC[C@@H](N)C3)-c3ccc(C#N)c(F)c3)c(F)cc12

InChI Key InChIKey=ITWXASOKPURBPP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 640925   

TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640925((R)-4-(8-(3-aminopiperidin-1-yl)-3-(6-fluoro-1-met...)
Affinity DataIC50: 1nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
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Date in BDB:
2/3/2024
Entry Details
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