BDBM639432 ({3- fluorobicyclo[1.1.1] pentan-1-yl}methyl) ({[2-({4-[5- (morpholin-4- yl)pyridin-3-yl]-1H- 1,2,3-triazol-1- yl}methyl)imidazo [1,2-a]pyridin-6- yl]methyl})amine::US20230391770, Example 52

SMILES FC12CC(CNCc3ccc4nc(Cn5cc(nn5)-c5cncc(c5)N5CCOCC5)cn4c3)(C1)C2

InChI Key InChIKey=GNOZRFWSLUASSE-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 639432   

TargetN6-adenosine-methyltransferase catalytic/non-catalytic subunit(Human)
Storm Therapeutics

US Patent

LigandBDBM639432(({3- fluorobicyclo[1.1.1] pentan-1-yl}methyl) ({[2...)Copy SMILESCopy InChI

Affinity DataIC50: 6nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
1/28/2024
Entry Details
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