BDBM639309 N-(2-fluoro-4-hydroxy- cyclohexyl)-7-[2-(2,2,2- trifluoroethoxy)phenyl] benzofuran-2-carboxamide::US20230391758, Compound 11

SMILES OC1CCC(NC(=O)c2cc3cccc(-c4ccccc4OCC(F)(F)F)c3o2)C(F)C1

InChI Key InChIKey=UXYRGWBJWCDHJI-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 639309   

TargetCeramide glucosyltransferase(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM639309(N-(2-fluoro-4-hydroxy- cyclohexyl)-7-[2-(2,2,2- tr...)
Affinity DataEC50:  7.10nMAssay Description:Using Promega's UDP-Glo™ Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2024
Entry Details
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