BDBM629038 3-(1-Methyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl)isothiazole;::US20230339900, Example 15

SMILES Cn1cc(c(n1)-c1ccsn1)-c1ccnc2[nH]ccc12

InChI Key InChIKey=UGKXDQUEXADBQG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 629038   

TargetCasein kinase I isoform delta(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM629038(US20230339900, Example 15 | 3-(1-Methyl-4-(1H-pyrr...)
Affinity DataIC50: 181nMAssay Description:In this assay, CSNK1D phosphorylates a substrate peptide PLSRTL-pS-VASLPGL in the presence of ATP. This substrate peptide has been modeled after the ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
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