BDBM626392 1-(1-(4-fluorophenyl)-6-methyl-1H-indazol-5-yl)-N-methyl-N-(1-propyl-1H-pyrazol-4-yl)pyrrolidine-3-sulfonamide::US11787780, Example 29

SMILES CCCn1cc(NS(=O)(=O)C2CCN(C2)c2cc3cnn(-c4ccc(F)cc4)c3cc2C)cn1

InChI Key InChIKey=XNXOPYUQETVKNC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 626392   

TargetGlucocorticoid receptor(Human)
Corcept Therapeutics

US Patent
LigandPNGBDBM626392(US11787780, Example 29 | 1-(1-(4-fluorophenyl)-6-m...)
Affinity DataIC50: 9nMAssay Description:Binding of test compounds to the glucocorticoid receptor (GR) is determined using a fluorescence polarisation (FP) assay utilising a recombinant liga...More data for this Ligand-Target Pair
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Date in BDB:
11/29/2023
Entry Details
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