BDBM625472 US20230322789, Compound 105::US20230322789, Example 72

SMILES CCS(=O)(=O)N1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F

InChI Key InChIKey=XRNIQXKGBKOKPT-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 625472   

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Broadenbio

US Patent

LigandBDBM625472(US20230322789, Compound 105 | US20230322789, Examp...)Copy SMILESCopy InChI

Affinity DataIC50: 50nMAssay Description:1. HPK1 Kinase Activity Inhibition Test. The kinase activity of HPK1 is manifested as activity of autophosphorylation and phosphorylation of downstre...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
11/22/2023
Entry Details
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