BDBM611494 (2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[6- (trifluoromethyl)-3- pyridyl]pyrimidin-4- yl]methyl]azetidine-2- carboxamide::US10626112, Example 388

SMILES Fc1ccc2oc(cc2c1)S(=O)(=O)N1CCC1C(=O)NCc1cc(ncn1)-c1ccc(nc1)C(F)(F)F

InChI Key InChIKey=GFMAGFPTNGJURF-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 611494   

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Ea Pharma

US Patent

LigandBDBM611494((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[6...)Copy SMILESCopy InChI

Affinity DataIC50: 2.70nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/8/2023
Entry Details
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