BDBM611396 (2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[2-hydroxy-4- (trifluoromethyl)phenyl]pyrimidin-4- yl]methyl]pyrrolidine-2-carboxamide::US10626112, Example 289

SMILES Oc1cc(ccc1-c1cc(CNC(=O)[C@@H]2CCCN2S(=O)(=O)c2cc3cc(F)ccc3o2)ncn1)C(F)(F)F

InChI Key InChIKey=PDXHELDREDKQCC-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 611396   

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Ea Pharma

US Patent

LigandBDBM611396((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[2...)Copy SMILESCopy InChI

Affinity DataIC50: 1.40nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/8/2023
Entry Details
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