BDBM611380 (2S)-1-furo[3,2-c]pyridin-2- ylsulfonyl-N-[[4-hydroxy-3- [5-(trifluoromethyl)-2- pyridyl]phenyl]methyl]- pyrrolidine-2-carboxamide::US10626112, Example 273

SMILES Oc1ccc(CNC(=O)[C@@H]2CCCN2S(=O)(=O)c2cc3cnccc3o2)cc1-c1ccc(cn1)C(F)(F)F

InChI Key InChIKey=RQSZRHYLICXZOY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 611380   

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Ea Pharma

US Patent

LigandBDBM611380((2S)-1-furo[3,2-c]pyridin-2- ylsulfonyl-N-[[4-hydr...)Copy SMILESCopy InChI

Affinity DataIC50: 1.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/8/2023
Entry Details
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