BDBM611365 (1R,3S,5R)-4-(5- fluorobenzofuran-2-yl)sulfonyl- N-[[4-[5-(trifluoromethyl)-2- pyridyl]-2-pyridyl]methyl]-4- azabicyclo[3.1.0]hexane-3- carboxamide::US10626112, Example 258

SMILES Fc1ccc2oc(cc2c1)S(=O)(=O)N1[C@@H]2C[C@@H]2C[C@H]1C(=O)NCc1cc(ccn1)-c1ccc(cn1)C(F)(F)F

InChI Key InChIKey=ROYZFBSQDCFUJI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 611365   

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Ea Pharma

US Patent

LigandBDBM611365((1R,3S,5R)-4-(5- fluorobenzofuran-2-yl)sulfonyl- N...)Copy SMILESCopy InChI

Affinity DataIC50: 1.90nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/8/2023
Entry Details
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