BDBM611230 (2S)-1-(benzofuran-2- ylsulfonyl)-N-[[2-[2-hydroxy-4- (trifluoromethyl)phenyl]-4- pyridyl]methyl]pyrrolidine-2- carboxamide::US10626112, Example 123

SMILES Oc1cc(ccc1-c1cc(CNC(=O)C2CCCN2S(=O)(=O)c2cc3ccccc3o2)ccn1)C(F)(F)F

InChI Key InChIKey=SAHFVTJLBQYSRR-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 611230   

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Ea Pharma

US Patent

LigandBDBM611230((2S)-1-(benzofuran-2- ylsulfonyl)-N-[[2-[2-hydroxy...)Copy SMILESCopy InChI

Affinity DataIC50: 2.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/8/2023
Entry Details
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