BDBM611147 (2S)-N-[(3-benzyloxy-5- fluoro-phenyl)methyl]- 1-(5-fluorobenzofuran- 2-yl)sulfonyl- pyrrolidine-2-carboxamide::US10626112, Example 34

SMILES Fc1cc(CNC(=O)[C@@H]2CCCN2S(=O)(=O)c2cc3cc(F)ccc3o2)cc(OCc2ccccc2)c1

InChI Key InChIKey=POMLHMWBBRGTOT-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 611147   

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Ea Pharma

US Patent

LigandBDBM611147((2S)-N-[(3-benzyloxy-5- fluoro-phenyl)methyl]- 1-(...)Copy SMILESCopy InChI

Affinity DataIC50: 1.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/8/2023
Entry Details
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