BDBM600479 US11622967, Example SUVN-G3031

SMILES O=C(CN1CCOCC1)Nc1ccc(OC2CCN(CC2)C2CCC2)cc1

InChI Key InChIKey=LNXDUSQEXVQFGP-UHFFFAOYSA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 600479   

TargetHistamine H3 receptor(Rat)
Suven Life Sciences

US Patent
LigandPNGBDBM600479(US11622967, Example SUVN-G3031)
Affinity DataIC50: 20nMAssay Description:Histamine-3 membranes were prepared from recombinant CHO-k1 cells expressing human histamine-3 receptor or rat histamine-3 receptor. Radioligand (RS)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2023
Entry Details
Go to US Patent

TargetHistamine H3 receptor(Human)
Suven Life Sciences

US Patent
LigandPNGBDBM600479(US11622967, Example SUVN-G3031)
Affinity DataKi:  8.73nMAssay Description:Histamine-3 membranes were prepared from recombinant CHO-k1 cells expressing human histamine-3 receptor or rat histamine-3 receptor. Radioligand (RS)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2023
Entry Details
Go to US Patent

TargetHistamine H3 receptor(Rat)
Suven Life Sciences

US Patent
LigandPNGBDBM600479(US11622967, Example SUVN-G3031)
Affinity DataKi:  9.79nMAssay Description:Histamine-3 membranes were prepared from recombinant CHO-k1 cells expressing human histamine-3 receptor or rat histamine-3 receptor. Radioligand (RS)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2023
Entry Details
Go to US Patent