BDBM595696 5-(2,4-Dimethyl-3-oxopiperazin-1-yl)-3-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazolo[4,3-b]pyridine-6-carbonitrile::US11591329, Ex. No. 23

SMILES CC1N(CCN(C)C1=O)c1nc2c(n[nH]c2cc1C#N)-c1cnn(C)c1

InChI Key InChIKey=QOWKYDUXRGQNEC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 595696   

TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595696(US11591329, Ex. No. 23 | 5-(2,4-Dimethyl-3-oxopipe...)
Affinity DataIC50: 115nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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